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CuBr-Promoted Tandem Cyclization/Trifluoromethylation of 2-Alkynylanilines: Efficient Synthesis of 3-Trifluoromethylindoles
Alternative TitleCuBr促进的邻炔苯胺串联环化三氟甲基化反应: 高效合成3-三氟甲基吲哚
Ge GC(葛广存); Huang XJ(黄小军); Ding CH(丁昌华); LI HAO; WAN SHILI; Hou XL(侯雪龙)
2014
Source PublicationChin. J. Chem.
Volume32Issue:8Pages:727-733
AbstractA new efficient strategy for the synthesis of 3-trifluoromethyl-indoles was developed through tandem cyclization/trifluoromethylation of 2-alkynylanilines and Umemoto's reagent under effect of CuBr. The reaction features the use of cheap copper salt, mild reaction conditions and high yield of products. The preliminary mechanism study indicates the solvent dimethylacetamide acts as the role of dealkylation.
Subject Area金属有机化学
DOI10.1002/cjoc.201400298
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Indexed BySCI
Language英语
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Cited Times:12[WOS]   [WOS Record]     [Related Records in WOS]
Document Type期刊论文
Identifierhttp://ir.sioc.ac.cn/handle/331003/39108
Collection金属有机化学国家重点实验室
Corresponding AuthorHou XL(侯雪龙)
Affiliation中科院上海有机化学研究所
Recommended Citation
GB/T 7714
Ge GC,Huang XJ,Ding CH,et al. CuBr-Promoted Tandem Cyclization/Trifluoromethylation of 2-Alkynylanilines: Efficient Synthesis of 3-Trifluoromethylindoles[J]. Chin. J. Chem.,2014,32(8):727-733.
APA 葛广存,黄小军,丁昌华,LI HAO,WAN SHILI,&侯雪龙.(2014).CuBr-Promoted Tandem Cyclization/Trifluoromethylation of 2-Alkynylanilines: Efficient Synthesis of 3-Trifluoromethylindoles.Chin. J. Chem.,32(8),727-733.
MLA 葛广存,et al."CuBr-Promoted Tandem Cyclization/Trifluoromethylation of 2-Alkynylanilines: Efficient Synthesis of 3-Trifluoromethylindoles".Chin. J. Chem. 32.8(2014):727-733.
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